SCHEMBL13869873

SCHEMBL13869873

CCCCC1CCCc2c1sc(NC(C)=O)c2C(=O)OCC

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.52
HTT P42858 2/20 0.52
MAPK1 P28482 2/20 0.52
GAA P10253 1/20 0.52
USP2 O75604 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
TSHR P16473 6/20 0.52
HPGD P15428 2/20 0.52
MAPT P10636 8/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 5/20 0.47
HSD17B10 Q99714 3/20 0.47
ALOX15 P16050 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 1/20 0.45
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13886696 0.83 CXCR2 (0.53) ALDH1A1GAATSHRMAPTSMN1; SMN2
SCHEMBL13869872 0.82 PDE4D (0.54) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL3987717 0.80 ALDH1A1 (0.56) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL3982213 0.77 ALDH1A1 (0.52) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL3990317 0.77 THRB (0.57) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL13886697 0.76 ALDH1A1 (0.48) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL2306161 0.74 MAPT (0.76) ALDH1A1GAATSHRHPGDMAPT
SCHEMBL13779376 0.74 ALDH1A1 (0.81) ALDH1A1GAATSHRHPGDMAPT
SCHEMBL3982274 0.74 ALDH1A1 (0.53) ALDH1A1HTTMAPK1GAAUSP2
SCHEMBL5484664 0.73 ALDH1A1 (0.50) ALDH1A1HTTMAPK1GAAUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7524853-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2009-04-28 US disclosed
US-7524853-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2009-04-28 US disclosed
US-7465739-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-16 US disclosed
US-7465739-B2 Compounds and their use in therapy SOLVAY PHARMACEUTICALS B.V. (NL) 2008-12-16 US disclosed