SCHEMBL1387206

SCHEMBL1387206

COc1cc2ncnc(Nc3ccc(Oc4ccccc4)cc3)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 1.00
RIPK2 O43353 2/20 1.00
EPHB2 P29323 1/20 1.00
KDR P35968 6/20 0.81
RET P07949 3/20 0.81
LCK P06239 5/20 0.79
SRC P12931 1/20 0.70
ERBB2 P04626 1/20 0.69
ERBB4 Q15303 1/20 0.69
FLT1 P17948 1/20 0.69
GAK O14976 1/20 0.69
STK10 O94804 1/20 0.69
FLT3 P36888 1/20 0.69
JAK3 P52333 1/20 0.69
AAK1 Q2M2I8 1/20 0.69
Q6ZSR9 Q6ZSR9 1/20 0.69
SLK Q9H2G2 1/20 0.69
IRAK4 Q9NWZ3 1/20 0.69
RPS6KA6 Q9UK32 1/20 0.69
ALK Q9UM73 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29385451 1.00 EGFR (1.00) EGFRRIPK2EPHB2KDRRET
Hydrochloric Acid SCHEMBL8807925 0.99 EGFR (0.98) EGFRRIPK2EPHB2KDRRET
SCHEMBL21442463 0.92 EGFR (0.84) EGFRRIPK2EPHB2KDRRET
SCHEMBL15390777 0.91 EGFR (0.83) EGFRRIPK2EPHB2KDRRET
SCHEMBL18158215 0.90 EGFR (0.82) EGFRRIPK2EPHB2KDRRET
SCHEMBL1387182 0.90 EGFR (0.94) EGFRRIPK2EPHB2KDRRET
SCHEMBL29515328 0.90 EGFR (1.00) EGFRRIPK2EPHB2KDRRET
SCHEMBL1257431 0.90 EGFR (1.00) EGFRRIPK2EPHB2KDRRET
Hydrochloric Acid SCHEMBL8811926 0.89 EGFR (0.80) EGFRRIPK2EPHB2KDRRET
SCHEMBL8933814 0.89 KDR (0.88) EGFRRIPK2EPHB2KDRRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 125 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11752150-B2 Anti-tumor immunotherapy enhancer NOBUO TSUKAMOTO (JP) 2023-09-12 US claimed
US-20200383981-A1 Anti-Tumor Immunotherapy Enhancer KEIO UNIVERSITY (JP) 2020-12-10 US claimed
US-20170172989-A1 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS BAYER HEALTHCARE LLC (US) 2017-06-22 US claimed
EP-2600150-B1 Method for determining sensitivity of tumor cells to dasatinib and computer program SYSMEX CORP (JP) 2015-01-07 EP claimed
US-20130143236-A1 METHOD FOR DETERMINING SENSITIVITY OF TUMOR CELLS TO DASATINIB AND COMPUTER PROGRAM SYSMEX CORPORATION (JP) 2013-06-06 US claimed
EP-2600150-A2 Method for determining sensitivity of tumor cells to dasatinib and computer program Sysmex Corporation (JP) 2013-06-05 EP claimed
EP-2400033-B1 Method for determining sensitivity of tumor cells to tyrosine kinase inhibitor and computer program product SYSMEX CORP (JP) 2013-02-20 EP claimed
US-20110318768-A1 METHOD FOR DETERMINING SENSITIVITY OF TUMOR CELLS TO TYROSINE KINASE INHIBITOR AND COMPUTER PROGRAM PRODUCT SYSMEX CORPORATION (JP) 2011-12-29 US claimed
EP-2400033-A1 Method for determining sensitivity of tumor cells to tyrosine kinase inhibitor and computer program product SYSMEX CORPORATION (JP) 2011-12-28 EP claimed
US-20100173954-A1 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS BAYER HEALTHCARE LLC (US) 2010-07-08 US claimed
EP-2114403-A2 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS Bayer Healthcare, LLC (US) 2009-11-11 EP claimed
WO-2008089388-A2 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS BAYER HEALTHCARE LLC (US) 2008-07-24 WO claimed
JP-H10505600-A 1998-06-02 JP claimed
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP claimed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO claimed
WO-2025261943-A1 ANTI-CANCER COMBINATIONS COMPRISING MOSPERAFENIB AND FOLFOX OR FOLFIRI F. HOFFMANN-LA ROCHE AG (CH) 2025-12-26 WO disclosed
EP-4634172-A1 COMBINATION THERAPY FOR CANCER TREATMENT F. Hoffmann-La Roche AG (CH) 2025-10-22 EP disclosed
WO-2004001384-A2 METHODS FOR INHIBITING ANGIOGENESIS, CELL MIGRATION, CELL ADHESION, AND CELL SURVIVAL THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2003-12-31 WO disclosed
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170172989-A1 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS CDK4, TP53, ABCC1 EGFR 411/4885RIPK2 2901/4885EPHB2 2830/4885
US-20100173954-A1 TREATMENT OF CANCERS HAVING RESISTANCE TO CHEMOTHERAPEUTIC AGENTS CDK4, TP53, ABCC1 EGFR 411/4885RIPK2 2901/4885EPHB2 2830/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.