SCHEMBL1387699

SCHEMBL1387699

CCSC(=N)Nc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.60
RAB9A P51151 5/20 0.58
NPC1 O15118 5/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C19 P33261 1/20 0.57
LTA4H P09960 2/20 0.55
NOX1 Q9Y5S8 2/20 0.54
NOS3 P29474 2/20 0.53
NOS1 P29475 2/20 0.53
NOS2 P35228 2/20 0.53
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
GPR55 Q9Y2T6 1/20 0.53
RECQL P46063 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387462 0.82 HPGD (0.54) ALDH1A1RAB9ANPC1SMN1; SMN2MEN1
Iodide SCHEMBL7787919 0.81 HPGD (0.52) ALDH1A1RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL4979973 0.81 MEN1 (0.69) ALDH1A1RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL1387773 0.80 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2KMT2ACYP2C19RECQL
Bromide SCHEMBL11804669 0.78 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KMT2ACYP2C19RECQL
Iodide SCHEMBL6699561 0.78 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KMT2ACYP2C19NOS3
SCHEMBL27479163 0.78 C5AR1 (0.47) ALDH1A1MEN1KMT2A
SCHEMBL4987199 0.78 LTA4H (0.66) ALDH1A1RAB9ANPC1SMN1; SMN2MEN1
SCHEMBL7787971 0.77 SMN1; SMN2 (0.50) ALDH1A1RAB9ANPC1SMN1; SMN2KMT2A
Hydrochloric Acid SCHEMBL27564382 0.77 C5AR1 (0.46) ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H09504278-A 1997-04-28 JP claimed
EP-0723438-A1 SUBSTITUTED UREA AND ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-31 EP claimed
WO-1995009619-A2 SUBSTITUTED UREA AND ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-04-13 WO claimed
US-6297276-B1 Substituted urea and isothiourea derivatives as no synthase inhibitors GLAXOSMITHKLINE 2001-10-02 US disclosed
US-6225305-B1 Substituted urea and isothiorea derivatives as no synthase inhibitors GLAXO WELLCOME INC. 2001-05-01 US disclosed
US-6090846-A ADMINISTERING S-ETHYL-N-((4-TRIFLUOROMETHYL)PHENYL)ISOTHIOUREA GLAXO WELLCOME INC. (US) 2000-07-18 US disclosed
EP-0723438-A1 SUBSTITUTED UREA AND ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-07-31 EP disclosed
WO-1995009619-A2 SUBSTITUTED UREA AND ISOTHIOUREA DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-04-13 WO disclosed