Iodide

Iodide

SCHEMBL6699561

CCSC(=N)Nc1ccccc1.I

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HDAC3 O15379 5/20 0.43
HDAC4 P56524 5/20 0.43
HDAC1 Q13547 5/20 0.43
HDAC7 Q8WUI4 5/20 0.43
HDAC2 Q92769 5/20 0.43
HDAC10 Q969S8 5/20 0.43
HDAC11 Q96DB2 5/20 0.43
HDAC8 Q9BY41 5/20 0.43
HDAC6 Q9UBN7 5/20 0.43
HDAC9 Q9UKV0 5/20 0.43
HDAC5 Q9UQL6 5/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
TAS2R38 P59533 1/20 0.41
NAPRT Q6XQN6 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387773 0.98 ALDH1A1 (0.46) ALDH1A1NPSR1HDAC3HDAC4HDAC1
Bromide SCHEMBL11804669 0.96 ALDH1A1 (0.45) ALDH1A1NPSR1HDAC3HDAC4HDAC1
Iodide SCHEMBL7787919 0.85 HPGD (0.52) ALDH1A1NPSR1SMN1; SMN2KMT2AGAA
SCHEMBL1387462 0.83 HPGD (0.54) ALDH1A1NPSR1SMN1; SMN2KMT2AGAA
SCHEMBL7788119 0.81 MAPT (0.44) ALDH1A1CYP2C19RECQLHSD17B10KMT2A
SCHEMBL1387536 0.81 POLB (0.47) ALDH1A1NOS3NOS1NOS2
Iodide SCHEMBL1286893 0.79 HSD17B10 (0.46) ALDH1A1SMN1; SMN2TAS2R38NAPRTHSD17B10
SCHEMBL1387416 0.79 RAB9A (0.45) ALDH1A1SMN1; SMN2HSD17B10NOS3NOS1
SCHEMBL7982053 0.79 HDAC3 (0.46) ALDH1A1NPSR1HDAC3HDAC4HDAC1
SCHEMBL1387586 0.79 NOS1 (0.46) ALDH1A1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116490-A1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2004-06-17 US disclosed
EP-1381360-A1 COMPOUNDS AND METHODS FOR INHIBITING METAP2 IN MAMMALS SmithKline Beecham Corporation (US) 2004-01-21 EP disclosed
WO-2002078697-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed
US-4056527-A HERBICIDE BAYER AKTIENGESELLSCHAFT (DT) 1977-11-01 US disclosed