SCHEMBL13891713

SCHEMBL13891713

CSc1nc2c(c(-c3ccccc3)n1)C(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CCCO2

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.42
GRIN1 Q05586 2/20 0.39
GRIN2B Q13224 2/20 0.39
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
ADRB2 P07550 1/20 0.35
FPR1 P21462 1/20 0.35
GPR183 P32249 1/20 0.35
APLNR P35414 1/20 0.35
GLP1R P43220 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35
GPR35 Q9HC97 1/20 0.35
TNIK Q9UKE5 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891760 0.89 TACR1 (0.41) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL13891758 0.86 TACR1 (0.41) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL13891704 0.84 PIK3R1 (0.46) TACR1
SCHEMBL13891737 0.84 TACR1 (0.41) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL5229260 0.83 TACR1 (0.41) TACR1ROCK2ROCK1ADRB2FPR1
SCHEMBL6790261 0.82 TACR1 (0.45) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL5530949 0.80 TACR1 (0.44) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL6794955 0.79 TACR1 (0.49) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL14514053 0.79 GRIN1 (0.40) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL13891738 0.78 TACR1 (0.41) TACR1GRIN1GRIN2BROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed