SCHEMBL13891737

SCHEMBL13891737

CSc1nc2c(c(-c3ccc(F)cc3C)n1)C(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CCCO2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.41
HSP90AB1 P08238 2/20 0.36
WDR5 P61964 5/20 0.36
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
TNIK Q9UKE5 2/20 0.34
GRIN1 Q05586 2/20 0.33
GRIN2B Q13224 2/20 0.33
P2RX7 Q99572 2/20 0.33
ADRB2 P07550 1/20 0.33
FPR1 P21462 1/20 0.33
GPR183 P32249 1/20 0.33
APLNR P35414 1/20 0.33
GLP1R P43220 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
GPR35 Q9HC97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891760 0.90 TACR1 (0.41) TACR1ROCK2ROCK1GRIN1GRIN2B
SCHEMBL13891759 0.87 TACR1 (0.37) TACR1WDR5ROCK2ROCK1TNIK
SCHEMBL13891758 0.84 TACR1 (0.41) TACR1ROCK2ROCK1GRIN1GRIN2B
SCHEMBL13891713 0.84 TACR1 (0.42) TACR1ROCK2ROCK1TNIKGRIN1
SCHEMBL13891686 0.78 MAPT (0.35) P2RX7
SCHEMBL13891705 0.78 MTOR (0.38) TACR1ROCK2ROCK1TNIKADRB2
SCHEMBL13891719 0.76 TACR1 (0.48) TACR1ROCK2ROCK1
SCHEMBL13891718 0.75 TACR1 (0.40) TACR1ROCK2ROCK1GRIN1GRIN2B
SCHEMBL13891738 0.75 TACR1 (0.41) TACR1ROCK2ROCK1TNIKGRIN1
SCHEMBL5229635 0.75 TACR1 (0.41) TACR1ADRB2FPR1GPR183APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed