SCHEMBL13891738

SCHEMBL13891738

CS(=O)(=O)c1nc2c(c(-c3ccc(F)cc3)n1)C(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)CCCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.41
KDM4E B2RXH2 1/20 0.37
MITF O75030 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
STAT3 P40763 1/20 0.37
STAT1 P42224 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TLR9 Q9NR96 1/20 0.37
GRIN1 Q05586 3/20 0.35
GRIN2B Q13224 3/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
TNIK Q9UKE5 2/20 0.33
PTGS2 P35354 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891759 0.89 TACR1 (0.37) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL13891702 0.85 KDM4E (0.41) TACR1KDM4EMITFALDH1A1LMNA
SCHEMBL5225857 0.84 TACR1 (0.40) TACR1KDM4EMITFALDH1A1LMNA
SCHEMBL13891619 0.83 MTOR (0.47) TACR1ALDH1A1LMNAMEN1CYP1A2
SCHEMBL13891616 0.80 SDHB (0.40) TACR1ROCK2ROCK1TNIKPTGS2
SCHEMBL5528780 0.79 TACR1 (0.38) TACR1ROCK2ROCK1TNIKMEN1
SCHEMBL5532454 0.79 TACR1 (0.41) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL13891713 0.78 TACR1 (0.42) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL5527548 0.77 ADRB2 (0.46) TACR1GRIN1GRIN2BROCK2ROCK1
SCHEMBL5228204 0.76 TACR1 (0.41) TACR1ALDH1A1LMNASTAT3STAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed