SCHEMBL13893237

SCHEMBL13893237

Cc1ncccc1-c1nc(-c2ccccc2F)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.48
NPC1 O15118 4/20 0.44
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
VHL P40337 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
HTR3A P46098 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
KDM5B Q9UGL1 1/20 0.37
IDO1 P14902 1/20 0.37
SCD O00767 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.36
MPL P40238 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28231982 0.79 KDM4E (0.50) TDO2NPC1VHLKDM4EGAA
SCHEMBL13141588 0.79 PDE5A (0.41) NPC1CASP3SENP8SENP7SENP6
SCHEMBL13141590 0.78 GABRG2 (0.43) TDO2NPC1CASP3SENP8SENP7
SCHEMBL27741609 0.76 MAP4K1 (0.46) NPC1CASP3SENP8SENP7SENP6
SCHEMBL11695271 0.75 TDO2 (0.46) TDO2VHL
SCHEMBL27741619 0.73 DCUN1D1 (0.45) NPC1CASP3SENP8SENP7SENP6
SCHEMBL8784700 0.73 GAA (0.47) NPC1L3MBTL1MGAMGAASI
SCHEMBL7372676 0.72 NPC1 (0.52) TDO2NPC1KDM4EGAARAB9A
SCHEMBL8629915 0.71 PDGFRB (0.36) NPC1CASP3SENP8SENP7SENP6
SCHEMBL29662748 0.71 CSNK1D (0.48) NPC1CASP3SENP8SENP7SENP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009051705-A1 SUBSTITUTED 1,2,4-OXADIAZOLES AND ANALOGS THEREOF AS CB2 RECEPTOR MODULATORS, USEFUL IN THE TREATMENT OF PAIN, RESPIRATORY AND NON-RESPIRATORY DISEASES MERCK & CO., INC. (US) 2009-04-23 WO disclosed