SCHEMBL13893955

SCHEMBL13893955

Cc1c(NC(=O)c2cc3ccccc3s2)cccc1-c1c[nH]c(=O)c(N)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHPS P49366 6/20 0.51
BTK Q06187 3/20 0.48
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 5/20 0.45
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
F10 P00742 1/20 0.42
TMIGD3 P0DMS9 2/20 0.41
ADORA1 P30542 2/20 0.41
STAT1 P42224 1/20 0.41
CASP3 P42574 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13893940 0.82 BTK (0.53) BTKALDH1A1LMNA
SCHEMBL13894283 0.78 BTK (0.53) BTKHDAC1HDAC2
SCHEMBL171471 0.78 BTK (0.67) DHPSBTKALDH1A1
SCHEMBL1038028 0.76 BTK (0.49) DHPSBTK
SCHEMBL13894036 0.75 ITK (0.54) BTKHDAC1ALDH1A1LMNA
SCHEMBL12663172 0.74 HDAC2 (0.70) DHPSHDAC1HDAC2HDAC3HDAC4
SCHEMBL105874 0.73 BTK (0.54) DHPSBTKHDAC1ALDH1A1LMNA
SCHEMBL13894035 0.73 TAS1R3 (0.50) HDAC1HDAC2
SCHEMBL171444 0.72 BTK (0.45) BTKALDH1A1LMNA
SCHEMBL30050486 0.71 HDAC2 (0.54) DHPSHDAC1HDAC2HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed