SCHEMBL13894283

SCHEMBL13894283

Cc1ccc(C(=O)Nc2cccc(-c3c[nH]c(=O)c(N)c3)c2C)cc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BTK Q06187 4/20 0.53
ITK Q08881 4/20 0.53
PARP1 P09874 1/20 0.50
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HDAC2 Q92769 1/20 0.42
HDAC1 Q13547 1/20 0.42
AURKA O14965 1/20 0.41
TTK P33981 1/20 0.41
AURKB Q96GD4 1/20 0.41
INCENP Q9NQS7 1/20 0.41
POLB P06746 1/20 0.41
KIT P10721 1/20 0.41
SRC P12931 1/20 0.41
FLT3 P36888 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171471 0.90 BTK (0.67) BTKITKNPC1RAB9APOLB
SCHEMBL13894036 0.89 ITK (0.54) BTKITKMAPTNPC1RAB9A
SCHEMBL13893949 0.85 ITK (0.57) BTKITKPARP1MAPTTP53
SCHEMBL171447 0.80 BTK (0.54) BTKITKMAPTNPC1RAB9A
SCHEMBL13893955 0.78 DHPS (0.51) BTKHDAC2HDAC1
SCHEMBL13894035 0.76 TAS1R3 (0.50) MAPTNPC1RAB9AHDAC2HDAC1
SCHEMBL13893940 0.76 BTK (0.53) BTKMAPTNPC1RAB9APOLB
SCHEMBL13894290 0.75 ITK (0.58) BTKITKAURKATTKAURKB
SCHEMBL3870962 0.74 BTK (0.70) BTKITKNPC1RAB9APOLB
SCHEMBL171935 0.72 BTK (0.59) BTKITKNPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed