SCHEMBL13894285

SCHEMBL13894285

CNC(=O)Nc1cc(-c2cccc(-n3cnc4cc(C)ccc4c3=O)c2C)c[nH]c1=O

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BTK Q06187 19/20 0.61
ITK Q08881 2/20 0.39
JAK2 O60674 1/20 0.39
NTRK1 P04629 1/20 0.39
LCK P06239 1/20 0.39
LYN P07948 1/20 0.39
RET P07949 1/20 0.39
SRC P12931 1/20 0.39
TEC P42680 1/20 0.39
TXK P42681 1/20 0.39
BLK P51451 1/20 0.39
BMX P51813 1/20 0.39
KCNH2 Q12809 1/20 0.39
ERBB4 Q15303 1/20 0.39
NTRK2 Q16620 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108070 0.76 BTK (1.00) BTKITKJAK2NTRK1LCK
SCHEMBL8735247 0.76 BTK (0.76) BTKJAK2
SCHEMBL13893949 0.71 ITK (0.57) BTKITKSRC
SCHEMBL13894298 0.66 ITK (0.45) BTKITKSRC
SCHEMBL13894290 0.65 ITK (0.58) BTKITKSRCBMX
SCHEMBL13894037 0.65 ITK (0.50) BTKITKSRCKCNH2
SCHEMBL17699541 0.64 BTK (1.00) BTKITKJAK2NTRK1LCK
SCHEMBL29782619 0.64 BTK (1.00) BTKITKJAK2NTRK1LCK
SCHEMBL13894019 0.64 KDM4E (0.40) BTKJAK2
SCHEMBL13894049 0.63 BTK (0.43) BTKITKSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed