SCHEMBL13894290

SCHEMBL13894290

CNC(=O)Nc1cc(-c2cccc(NC(=O)c3ccc(N(C)C)cc3)c2C)c[nH]c1=O

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITK Q08881 9/20 0.58
KIT P10721 4/20 0.58
SRC P12931 4/20 0.58
FLT3 P36888 4/20 0.58
BTK Q06187 8/20 0.47
TTK P33981 2/20 0.43
AURKA O14965 1/20 0.43
AURKB Q96GD4 1/20 0.43
INCENP Q9NQS7 1/20 0.43
EGFR P00533 1/20 0.41
BMX P51813 1/20 0.41
JAK3 P52333 1/20 0.41
KCNK3 O14649 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13893949 0.90 ITK (0.57) ITKKITSRCFLT3BTK
SCHEMBL13894298 0.86 ITK (0.45) ITKKITSRCFLT3BTK
SCHEMBL13894036 0.86 ITK (0.54) ITKKITSRCFLT3BTK
SCHEMBL13894052 0.83 ITK (0.47) ITKKITSRCFLT3BTK
SCHEMBL106046 0.82 BTK (0.64) BTKEGFRBMXJAK3
SCHEMBL13894049 0.80 BTK (0.43) ITKKITSRCFLT3BTK
SCHEMBL13894122 0.79 ITK (0.54) ITKKITSRCFLT3BTK
SCHEMBL13894037 0.78 ITK (0.50) ITKKITSRCFLT3BTK
SCHEMBL3870962 0.77 BTK (0.70) ITKKITSRCFLT3BTK
SCHEMBL4080570 0.77 BTK (0.52) ITKKITSRCFLT3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed