SCHEMBL13894049

SCHEMBL13894049

CNC(=O)Nc1cc(-c2cccc(NC(=O)c3ccc4c(ccn4C)c3)c2C)c[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 3/20 0.43
ITK Q08881 10/20 0.42
MAOB P27338 1/20 0.41
SRC P12931 6/20 0.40
FLT3 P36888 6/20 0.40
KIT P10721 5/20 0.40
TTK P33981 3/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
AURKA O14965 2/20 0.37
AURKB Q96GD4 2/20 0.37
INCENP Q9NQS7 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108970 0.86 BTK (0.59) BTKMAOBKDM4EALDH1A1CYP1A2
SCHEMBL13893949 0.83 ITK (0.57) BTKITKSRCFLT3KIT
SCHEMBL13894290 0.80 ITK (0.58) BTKITKSRCFLT3KIT
SCHEMBL13894052 0.77 ITK (0.47) BTKITKSRCFLT3KIT
SCHEMBL13894298 0.77 ITK (0.45) BTKITKSRCFLT3KIT
SCHEMBL13894037 0.75 ITK (0.50) BTKITKSRCFLT3KIT
SCHEMBL3870962 0.71 BTK (0.70) BTKITKSRCFLT3KIT
SCHEMBL171935 0.70 BTK (0.59) BTKITKSRCFLT3KIT
SCHEMBL171856 0.70 HDAC3 (0.42) BTKMAOBHDAC3HDAC1AURKA
SCHEMBL13894283 0.69 BTK (0.53) BTKITKSRCFLT3KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed