SCHEMBL13905596

SCHEMBL13905596

CCOP(=O)(O)CN(c1ccc2cc(N)ccc2c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.34
HCRTR2 O43614 1/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 2/20 0.33
CNR2 P34972 2/20 0.32
ESR1 P03372 2/20 0.32
CNR1 P21554 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
PGR P06401 1/20 0.30
POLB P06746 1/20 0.30
BCL2L1 Q07817 2/20 0.30
MCL1 Q07820 2/20 0.30
HTR1A P08908 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR7 P34969 1/20 0.30
DRD3 P35462 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2055449 0.90 S1PR1 (0.35) S1PR1HCRTR2MAPTLMNACNR2
SCHEMBL3058248 0.86 S1PR1 (0.38) S1PR1HCRTR2PGRBCL2L1MCL1
SCHEMBL10292752 0.82 PER2 (0.37) S1PR1HCRTR2MAPTLMNA
SCHEMBL10291699 0.79 HCRTR2 (0.34) S1PR1HCRTR2KEAP1NFE2L2
SCHEMBL10291700 0.79 TAS1R3 (0.35) S1PR1HCRTR2LMNAPOLB
SCHEMBL10292014 0.78 ALDH1A1 (0.40) MAPTLMNA
SCHEMBL10292760 0.78 ALDH1A1 (0.44) HCRTR2MAPTLMNAPOLB
SCHEMBL10291993 0.77 ALDH1A1 (0.38) S1PR1MAPTPOLB
SCHEMBL2099883 0.75 S1PR1 (0.31) S1PR1
SCHEMBL13658664 0.75 PSEN1 (0.38) S1PR1HCRTR2MAPTKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed