SCHEMBL13939596

SCHEMBL13939596

CNC1CCN(S(=O)(=O)C2CC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.46
SMYD3 Q9H7B4 8/20 0.38
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TP53 P04637 1/20 0.32
JAK1 P23458 1/20 0.32
CCND1 P24385 2/20 0.32
CCNE1 P24864 2/20 0.32
CDK2 P24941 2/20 0.32
CDK6 Q00534 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8342421 0.92 EPHX2 (0.51) EPHX2SMYD3TSHRL3MBTL1
SCHEMBL23564023 0.88 EPHX2 (0.40) EPHX2SMYD3TSHRL3MBTL1TP53
SCHEMBL6118668 0.80 EPHX2 (0.47) EPHX2SMYD3TSHRL3MBTL1JAK1
SCHEMBL5344959 0.80 TP53 (0.50) EPHX2SMYD3TSHRL3MBTL1TP53
SCHEMBL9034989 0.80 CA1 (0.42) EPHX2SMYD3TSHRL3MBTL1TP53
SCHEMBL8978497 0.78 L3MBTL1 (0.53) EPHX2SMYD3TSHRL3MBTL1TP53
SCHEMBL14037777 0.76 EPHX2 (0.41) EPHX2SMYD3TSHRL3MBTL1
SCHEMBL8978496 0.75 ALDH1A1 (0.55) CCNE1CDK2
SCHEMBL14618813 0.75 EPHX2 (0.51) EPHX2TSHRL3MBTL1JAK1CCND1
SCHEMBL23973911 0.75 ADH1B (0.50) EPHX2SMYD3JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016460-A2 PYRAZOLE COMPOUNDS AND THEIR USE AS RAF INHIBITORS PFIZER INC. (US) 2009-02-05 WO disclosed