SCHEMBL13961453

SCHEMBL13961453

COBN1CCN(c2ccncc2NC(=O)c2ccnc(-c3ccc(Oc4ccccc4)cc3)n2)CC1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.56
GSK3B P49841 7/20 0.47
GSK3A P49840 6/20 0.47
PIM2 Q9P1W9 4/20 0.42
PRKCA P17252 2/20 0.42
PRKCQ Q04759 2/20 0.42
DYRK1A Q13627 4/20 0.41
PIM1 P11309 3/20 0.40
PIM3 Q86V86 3/20 0.40
MAPT P10636 1/20 0.40
ATR Q13535 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13961448 0.92 GSK3B (0.50) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961465 0.88 GSK3A (0.48) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961709 0.87 GSK3B (0.46) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961607 0.87 GSK3B (0.46) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961445 0.86 WDR5 (0.45) CHEK1GSK3BGSK3APIM2PIM1
SCHEMBL13028286 0.86 CHEK1 (0.55) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13028331 0.86 CHEK1 (0.72) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961466 0.85 PIM2 (0.47) GSK3BGSK3APIM2MAPT
SCHEMBL13961713 0.85 PIM2 (0.48) CHEK1GSK3BGSK3APIM2PRKCA
SCHEMBL13961456 0.84 GSK3B (0.47) CHEK1GSK3BGSK3APIM2PRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009014637-A2 HETEROCYCLIC AMIDE COMPOUNDS AS PROTEIN KINASE INHIBITORS SCHERING CORPORATION (US) 2009-01-29 WO disclosed