SCHEMBL1396210

SCHEMBL1396210

O=C1c2ccccc2C(=O)N1c1cc(O)[nH]n1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
ALPL P05186 4/20 0.40
ESR1 P03372 1/20 0.40
PIM3 Q86V86 1/20 0.40
HIPK4 Q8NE63 1/20 0.40
SCN2A Q99250 1/20 0.40
LMNA P02545 1/20 0.38
NR1H3 Q13133 3/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
PMP22 Q01453 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30645638 0.79 ALDH1A1 (0.44) ALDH1A1ALPLLMNAKDM4EGAA
SCHEMBL2113726 0.79 MEN1 (0.45) ALDH1A1ALPLKDM4EGAA
SCHEMBL17627048 0.79 ALDH1A1 (0.44) ALDH1A1ALPLLMNAKDM4EGAA
SCHEMBL16479224 0.76 ALOX15 (0.51) ALDH1A1ALPLLMNANR1H3HTT
SCHEMBL30475298 0.76 ALDH1A1 (0.41) ALDH1A1ALPLGAA
SCHEMBL3051213 0.76 ALDH1A1 (0.41) ALDH1A1ALPLGAA
SCHEMBL14858215 0.74 CCNA2 (0.42) ALDH1A1ALPL
SCHEMBL3996867 0.74 ALDH1A1 (0.45) ALDH1A1ALPLESR1PIM3HIPK4
SCHEMBL31727467 0.74 ALDH1A1 (0.45) ALDH1A1ALPLESR1PIM3HIPK4
SCHEMBL20582184 0.72 ALDH1A1 (0.38) ALDH1A1ALPLLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114945571-B Cyclic compounds and methods of use thereof 薛定谔公司 2025-02-25 CN disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2024-01-18 US disclosed
EP-4081526-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME Schrödinger, Inc. (US) 2022-11-02 EP disclosed
CN-114945571-A Cyclic compounds and methods of use thereof 薛定谔公司 2022-08-26 CN disclosed
WO-2021134004-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRODINGER, INC. (US) 2021-07-01 WO disclosed
WO-2021134004-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRODINGER, INC. (US) 2021-07-01 WO disclosed
US-20130165445-A1 Aurora Kinase Modulators and Method of Use AMGEN INC. (US) 2013-06-27 US disclosed
EP-2288611-B1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC (US) 2013-05-15 EP disclosed
US-8404694-B2 Aurora kinase modulators and method of use AMGEN INC. (US) 2013-03-26 US disclosed
US-20110065709-A1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC. (US) 2011-03-17 US disclosed
EP-2288611-A1 AURORA KINASE MODULATORS AND METHOD OF USE Amgen Inc. (US) 2011-03-02 EP disclosed
WO-2009117157-A1 AURORA KINASE MODULATORS AND METHOD OF USE AMGEN INC. (US) 2009-09-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110065709-A1 AURORA KINASE MODULATORS AND METHOD OF USE AURKC, AURKA, AURKB ALDH1A1 2417/4885ALPL 1450/4885ESR1 995/4885
US-20130165445-A1 Aurora Kinase Modulators and Method of Use AURKC, AURKA, AURKB ALDH1A1 2417/4885ALPL 1450/4885ESR1 995/4885
US-20240018157-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME MALT1, FKBP1B, FKBP1A ALDH1A1 2190/4885ALPL 3272/4885ESR1 4729/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.