SCHEMBL13986943

SCHEMBL13986943

O=C(N[C@H]1CCCCNC1=O)c1cc(-c2ccncc2)n[nH]c1=O

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.52
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
CHEK1 O14757 1/20 0.47
GSK3B P49841 1/20 0.47
CCR2 P41597 5/20 0.45
BDKRB1 P46663 1/20 0.44
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
KDM1A O60341 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14348304 1.00 ALDH1A1 (0.53) ALDH1A1KDM4ERAB9ANPC1CHEK1
SCHEMBL5236116 0.84 GSK3B (0.52) ALDH1A1CHEK1GSK3BMKNK2ROCK2
SCHEMBL4848283 0.83 GSK3B (0.51) ALDH1A1KDM4EGSK3BMKNK2ROCK2
SCHEMBL5233639 0.82 GSK3B (0.52) ALDH1A1CHEK1GSK3BMKNK1MKNK2
SCHEMBL5232508 0.82 MAPK8 (0.55) GSK3BMKNK1MKNK2ROCK2
SCHEMBL13987020 0.80 GSK3B (0.48) ALDH1A1KDM4EGSK3BMKNK1MKNK2
SCHEMBL14348317 0.78 GSK3B (0.45) ALDH1A1RAB9ANPC1GSK3BBDKRB1
SCHEMBL13986936 0.78 MAPK8 (0.51) ALDH1A1KDM4EGSK3BMKNK1MKNK2
SCHEMBL4854586 0.77 ROCK2 (0.52) ALDH1A1RAB9ANPC1GSK3BROCK2
SCHEMBL13986968 0.77 MAPK8 (0.50) RAB9ANPC1GSK3BROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7462613-B2 Pyridazinone derivatives as pharmaceuticals and pharmaceutical compositions containing them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-12-09 US disclosed
US-7462613-B2 Pyridazinone derivatives as pharmaceuticals and pharmaceutical compositions containing them SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-12-09 US disclosed