SCHEMBL13989449

SCHEMBL13989449

CN(C)CC12C=CC(C)(O1)[C@H]1C(=O)N(c3ccc(C#N)c(CF)c3)C(=O)[C@H]12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 12/20 0.44
CACNA1B Q00975 7/20 0.40
APBA1 Q02410 7/20 0.40
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
HSD17B10 Q99714 2/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13889592 0.88 CACNA1B (0.52) ARCACNA1BAPBA1ALDH1A1TP53
SCHEMBL13481656 0.85 AR (0.58) AR
SCHEMBL13889352 0.85 CACNA1B (0.43) ARCACNA1BAPBA1ALDH1A1TP53
SCHEMBL13889600 0.80 CACNA1B (0.46) ARCACNA1BAPBA1ALDH1A1TP53
SCHEMBL13989418 0.78 AR (0.53) ARCACNA1BAPBA1
SCHEMBL13889764 0.78 AR (0.54) ARCACNA1BAPBA1
SCHEMBL13989372 0.76 ALDH1A1 (0.37) ARCACNA1BAPBA1ALDH1A1TP53
SCHEMBL13889850 0.75 AR (0.74) ARCACNA1BAPBA1
SCHEMBL13482705 0.74 AR (0.49) AR
SCHEMBL13989444 0.74 AR (0.44) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470797-B2 Fused heterocyclic imido and amido compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-30 US disclosed