SCHEMBL14013777

SCHEMBL14013777

O=C1c2ccc(CO)cc2CCC1C(=O)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 8/20 0.42
S1PR1 P21453 1/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
CYP24A1 Q07973 2/20 0.37
CYP19A1 P11511 1/20 0.36
AKR1B1 P15121 1/20 0.35
CYP27A1 Q02318 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
GRIN2B Q13224 1/20 0.33
PDK2 Q15119 1/20 0.33
NAMPT P43490 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343955 0.82 PARP10 (0.40) CYP26A1CYP24A1CYP27A1
SCHEMBL4098450 0.79 CYP24A1 (0.54) CYP26A1CYP24A1CYP19A1CYP27A1DRD2
SCHEMBL6352009 0.79 ACHE (0.47) CYP19A1DRD2HTR2AHTR2CHTR2B
SCHEMBL29365032 0.79 ACHE (0.47) CYP19A1DRD2HTR2AHTR2CHTR2B
SCHEMBL18845473 0.71 CYP19A1 (0.49) CYP26A1CYP24A1CYP19A1CYP27A1GRIN2B
SCHEMBL10333984 0.71 CYP19A1 (0.48) CYP26A1CYP24A1CYP19A1CYP27A1
SCHEMBL6341940 0.69 HTR2C (0.39) HTR2C
SCHEMBL14013291 0.68 MAPT (0.53) CYP26A1CYP4F2CYP4A11CYP24A1CYP27A1
SCHEMBL7127913 0.68 AKR1B1 (0.42) S1PR1CYP4F2CYP4A11AKR1B1GRIN2B
SCHEMBL4805957 0.68 CASP1 (0.53) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed