SCHEMBL14017444

SCHEMBL14017444

CN1[C@@H]2CC[C@H]1C[C@H](Nc1ccccc1O)C2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.60
HTR3E A5X5Y0 1/20 0.60
HTR3B O95264 1/20 0.60
CHRM4 P08173 1/20 0.60
CHRM5 P08912 1/20 0.60
CHRNB2 P17787 1/20 0.60
CHRNB4 P30926 1/20 0.60
CHRNA3 P32297 1/20 0.60
HRH1 P35367 1/20 0.60
CHRNA7 P36544 1/20 0.60
CHRNA4 P43681 1/20 0.60
TMEM97 Q5BJF2 1/20 0.60
HTR3D Q70Z44 1/20 0.60
HTR3C Q8WXA8 1/20 0.60
SIGMAR1 Q99720 1/20 0.60
SLC6A2 P23975 4/20 0.45
SLC6A3 Q01959 1/20 0.45
KAT2B Q92831 1/20 0.45
CHRM1 P11229 3/20 0.43
SLC6A4 P31645 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3177266 1.00 HTR3A (0.60) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL6888233 0.94 HTR3A (0.69) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL6887110 0.94 HTR3A (0.69) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL13529096 0.80 HTR3E (0.46) HTR3AHTR3EHTR3BCHRM4CHRM5
Hydrochloric Acid SCHEMBL10538915 0.79 MEN1 (0.48) HTR3AMEN1KMT2AALDH1A1CYP3A4
SCHEMBL11104244 0.77 POLB (0.47) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL28306051 0.77 IDO1 (0.50) MEN1KMT2AALDH1A1CYP3A4HSD17B10
SCHEMBL6892215 0.76 CHRNA3 (0.71) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL6886540 0.76 CHRNA3 (0.71) HTR3AHTR3EHTR3BCHRM4CHRM5
SCHEMBL14191714 0.76 CHEK2 (0.39) HTR3AHTR3EHTR3BCHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439239-B2 Tricyclic δ- opioid modulators JANSSEN PHARMACEUTICA N.V. (BG) 2008-10-21 US disclosed
US-7439239-B2 Tricyclic δ- opioid modulators JANSSEN PHARMACEUTICA N.V. (BG) 2008-10-21 US disclosed