SCHEMBL14017684

SCHEMBL14017684

O=C(CO)N1CCC(N2CCC(O)CC2)CC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ACACB O00763 1/20 0.42
ACACA Q13085 1/20 0.42
CHRM1 P11229 1/20 0.40
ACHE P22303 4/20 0.39
L3MBTL3 Q96JM7 7/20 0.39
L3MBTL1 Q9Y468 6/20 0.39
MBTD1 Q05BQ5 4/20 0.39
TP53BP1 Q12888 2/20 0.39
L3MBTL4 Q8NA19 1/20 0.39
CYP2C19 P33261 2/20 0.38
KDM4E B2RXH2 2/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2D6 P10635 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1713072 0.88 ALDH1A1 (0.42) MEN1KMT2ACHRM1ALDH1A1
SCHEMBL13772727 0.83 MEN1 (0.58) MEN1KMT2AACHEL3MBTL3L3MBTL1
SCHEMBL13772749 0.83 MEN1 (0.58) MEN1KMT2AACHEL3MBTL3L3MBTL1
SCHEMBL13772800 0.80 L3MBTL3 (0.43) MEN1KMT2AACACBACACAACHE
SCHEMBL4720502 0.79 L3MBTL3 (0.42) MEN1KMT2ACHRM1L3MBTL3L3MBTL1
SCHEMBL13772828 0.78 KDM4E (0.50) MEN1KMT2AACHEL3MBTL3L3MBTL1
SCHEMBL13665501 0.76 DPP4 (0.49) CHRM1ALDH1A1
SCHEMBL1712955 0.76 DPP4 (0.49) CHRM1ALDH1A1
SCHEMBL13772875 0.75 L3MBTL3 (0.44) MEN1KMT2AACHEL3MBTL3L3MBTL1
SCHEMBL8353063 0.74 CHRM1 (0.70) CHRM1L3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863791-B1 2-OXO-1,2,4,5-TETRAHYDRO-1,3-BENZODIAZEPIN-3-YL-PIPERIDINES USED AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2008-11-12 EP disclosed