SCHEMBL14019207

SCHEMBL14019207

NC(=S)NNC(=O)c1cccc(F)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.67
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
PARP1 P09874 1/20 0.58
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
LMNA P02545 2/20 0.57
PKM P14618 1/20 0.57
HTT P42858 1/20 0.56
CTSL P07711 1/20 0.54
GAA P10253 2/20 0.52
KAT6A Q92794 1/20 0.52
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
CA1 P00915 1/20 0.51
CA9 Q16790 1/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8762392 0.81 LMNA (0.65) SMN1; SMN2NPC1RAB9AHDAC1HDAC6
SCHEMBL14907949 0.80 SMN1; SMN2 (1.00) SMN1; SMN2NPC1RAB9APARP1ALDH1A1
SCHEMBL8631029 0.80 NPC1 (0.58) SMN1; SMN2NPC1RAB9AHDAC1HDAC6
SCHEMBL20528632 0.79 CA1 (0.62) SMN1; SMN2RAB9AKDM4EALDH1A1GAA
SCHEMBL37273 0.78 ALDH1A1 (0.68) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL27860725 0.77 HDAC1 (0.65) SMN1; SMN2NPC1RAB9AHDAC1HDAC6
SCHEMBL405785 0.77 HDAC1 (0.69) NPC1RAB9AHDAC1HDAC6PARP1
SCHEMBL30046370 0.77 HDAC1 (0.69) NPC1RAB9AHDAC1HDAC6PARP1
SCHEMBL19672737 0.76 NPC1 (0.56) SMN1; SMN2NPC1RAB9AHDAC1HDAC6
SCHEMBL27163388 0.75 NPC1 (0.57) SMN1; SMN2NPC1RAB9AHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343503-B1 HETEROARYL UREA NEUROPEPTIDE Y Y5 RECEPTOR ANTAGONISTS SCHERING CORP (US) 2008-11-12 EP disclosed
US-7309704-B2 Heteroaryl urea neuropeptide Y Y5 receptor antagonists SCHERING CORPORATION (US) 2007-12-18 US disclosed
US-7309704-B2 Heteroaryl urea neuropeptide Y Y5 receptor antagonists SCHERING CORPORATION (US) 2007-12-18 US disclosed