SCHEMBL14023403

SCHEMBL14023403

CN(C)CC(C)(C)CNC(=O)c1cc(N)cc(Br)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
SLC6A5 Q9Y345 1/20 0.36
KCNA5 P22460 1/20 0.35
TP53BP1 Q12888 1/20 0.34
DDR1 Q08345 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR2 P34972 2/20 0.34
AKR1C3 P42330 2/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3542006 0.79 EPHX2 (0.51) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL14023398 0.78 ALDH1A1 (0.52) KDM4EALDH1A1CYP2C19GAASIGMAR1
SCHEMBL23139634 0.77 KDM4E (0.52) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL14334458 0.74 KDM4E (1.00) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL23786329 0.74 KDM4E (0.46) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL3543155 0.73 CYP2D6 (0.52) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL14500184 0.72 NPC1 (0.50) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL3541043 0.71 HTR4 (0.45) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL3115266 0.71 KDM4E (0.48) KDM4EALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL15485079 0.71 MEN1 (0.57) KDM4EALDH1A1MEN1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140420-A2 PYRIMIDINE DERIVATIVES S*BIO PTE LTD (SG) 2008-11-20 WO disclosed