SCHEMBL14040992

SCHEMBL14040992

COc1c(C)ccc2c1OCCO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2C P18825 2/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
ADRA2B P18089 1/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
PKM P14618 1/20 0.35
LMNA P02545 2/20 0.34
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10430779 0.85 POLB (0.43) HTT
SCHEMBL15988656 0.77 SMN1; SMN2 (0.41) SMN1; SMN2ALDH1A1KDM4EHPGDHTT
SCHEMBL13902883 0.75 ADRA2A (0.46) SMN1; SMN2ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL12446380 0.75 ALDH1A1 (0.40) SMN1; SMN2ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL14405280 0.74 HTR2C (0.37) SMN1; SMN2ADRA2AADRA2CADRA1A
SCHEMBL4714664 0.74 KDM4E (0.58) SMN1; SMN2ALDH1A1KDM4EHSD17B10HPGD
SCHEMBL14382047 0.73 CYP2A6 (0.38) KDM4ECTNNB1WNT3AADRA1DADRA1A
SCHEMBL19346092 0.73 SMN1; SMN2 (0.42) SMN1; SMN2ALDH1A1KDM4EHPGDHTT
SCHEMBL15988786 0.73 KDM4E (0.55) SMN1; SMN2ALDH1A1KDM4EHSD17B10CTNNB1
SCHEMBL30200165 0.73 KDM4E (0.55) SMN1; SMN2ALDH1A1KDM4EHSD17B10CTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1373257-B9 INHIBITORS OF C-JUN N-TERMINAL KINASES (JNK) AND OTHER PROTEIN KINASES VERTEX PHARMA (US) 2008-10-15 EP disclosed
EP-1373257-B1 INHIBITORS OF C-JUN N-TERMINAL KINASES (JNK) AND OTHER PROTEIN KINASES VERTEX PHARMA (US) 2007-11-28 EP disclosed