SCHEMBL14048520

SCHEMBL14048520

COC(=O)[C@@H]1C[C@H]1CN1CCC(c2csc3cc(C(F)(F)F)ccc23)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.41
DRD2 P14416 1/20 0.38
SLC6A4 P31645 1/20 0.38
CHRM4 P08173 1/20 0.36
HRH2 P25021 1/20 0.35
CYP3A4 P08684 2/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
KCNH2 Q12809 1/20 0.34
PPARD Q03181 3/20 0.33
PPARA Q07869 3/20 0.33
PPARG P37231 2/20 0.33
TRPV4 Q9HBA0 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
PTK2 Q05397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201192 0.89 CTSS (0.42) CTSSDRD2SLC6A4CHRM4HRH2
SCHEMBL2955859 0.84 ADRA1A (0.38) CHRM4CYP3A4MAPT
SCHEMBL2955868 0.84 ADRA1A (0.38) CHRM4CYP3A4MAPT
SCHEMBL2957073 0.84 ADRA1A (0.38) CHRM4CYP3A4MAPT
SCHEMBL2955865 0.84 ADRA1A (0.38) CHRM4CYP3A4MAPT
SCHEMBL2957077 0.84 ADRA1A (0.38) CHRM4CYP3A4MAPT
SCHEMBL2959717 0.80 CTSS (0.42) CTSSDRD2SLC6A4CHRM4TRPV1
SCHEMBL2957527 0.75 OPRD1 (0.37) CTSSKCNH2
SCHEMBL13221063 0.75 CTSS (0.38) CTSSDRD2SLC6A4CHRM4CYP3A4
SCHEMBL5022610 0.75 CTSS (0.36) CTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1632483-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2008-10-29 EP disclosed