SCHEMBL1408772

SCHEMBL1408772

O=C(Cl)OCC(Cl)(Cl)Cl.O=C(O)Cl

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
TP53 P04637 1/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28182083 0.95 ALDH1A1 (0.34) ALDH1A1CHRM2CHRM4CHRM1CHRM3
SCHEMBL3023 0.95
SCHEMBL41347 0.78
SCHEMBL28182085 0.77 CHRM2 (0.31) CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL4386155 0.76 ALDH1A1 (0.33) ALDH1A1CHRM2CHRM4CHRM1CHRM3
SCHEMBL236721 0.75 CHRM2 (0.37) ALDH1A1CHRM2CHRM4CHRM1CHRM3
SCHEMBL9230930 0.75 ALDH1A1 (0.34) ALDH1A1CHRM2CHRM4CHRM1CHRM3
SCHEMBL6660567 0.75 MAPK1 (0.39) ALDH1A1TP53
Clorethate SCHEMBL41346 0.75 CHRM2 (0.39) ALDH1A1CHRM2CHRM4CHRM1CHRM3
SCHEMBL9230926 0.74 ALDH1A1 (0.32) ALDH1A1TP53TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2294067-B1 PREPARATION OF N-6 DEMETHYLATED, 9-10-DIHYDROLYSERGIC ACID ALKYL ESTERS LEK PHARMACEUTICALS (SI) 2015-02-18 EP disclosed
EP-2294067-A1 PREPARATION OF N-6 DEMETHYLATED, 9-10-DIHYDROLYSERGIC ACID ALKYL ESTERS LEK Pharmaceuticals d.d. (SI) 2011-03-16 EP disclosed
WO-2009133097-A1 PREPARATION OF N-6 DEMETHYLATED, 9-10-DIHYDROLYSERGIC ACID ALKYL ESTERS LEK PHARMACEUTICALS D.D. (SI) 2009-11-05 WO disclosed
EP-2113504-A1 Preparation of N-6 demethylated, 9,10-dihydrolysergic acid alkyl esters LEK Pharmaceuticals D.D. (SI) 2009-11-04 EP disclosed