SCHEMBL1409150

SCHEMBL1409150

O=C(CN1C(=O)[C@@H](NC(=O)c2ccccc2)CNC2=C1CCC=C2)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.38
NAAA Q02083 3/20 0.37
CASP1 P29466 3/20 0.36
CASP3 P42574 1/20 0.36
CASP8 Q14790 1/20 0.36
GLA P06280 2/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL647101 0.80 RIPK1 (0.46) CTSLNAAACASP1
SCHEMBL1409814 0.78 CASP1 (0.37) CASP1CASP3CASP8
SCHEMBL646039 0.72 CASP1 (0.50) CASP1
SCHEMBL1409492 0.72 GAA (0.35)
SCHEMBL645174 0.71 CASP1 (0.49) CASP1
SCHEMBL645106 0.70 CASP1 (0.52) CASP1
SCHEMBL13140087 0.69 RIPK1 (0.42) CTSLNAAAGLA
SCHEMBL648535 0.68 XIAP (0.48)
SCHEMBL644741 0.66 SCN9A (0.47) CTSLNAAA
SCHEMBL5712951 0.64 CCKBR (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295442-A2 Inhibitors of interleukin-1beta converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-16 EP disclosed