SCHEMBL14101839

SCHEMBL14101839

Cc1ncnn1-c1cc(F)ccc1CNN

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.33
CASP6 P55212 2/20 0.32
P2RX7 Q99572 5/20 0.32
GAA P10253 2/20 0.31
MAPK1 P28482 1/20 0.31
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA5 P31644 2/20 0.30
PDE2A O00408 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12646546 0.86 P2RX7 (0.34) P2RX7GAAPDE2AMEN1KMT2A
SCHEMBL51809 0.85 MAPK14 (0.33) ATRP2RX7MAPK1GABRG2GABRB3
Hydrochloric Acid SCHEMBL2529209 0.83 MAPK14 (0.33) ATRP2RX7GABRG2GABRB3GABRA5
Hydrochloric Acid SCHEMBL2076893 0.83 MAPK14 (0.33) ATRP2RX7GABRG2GABRB3GABRA5
SCHEMBL12238979 0.74 GABRG2 (0.34) ATRGAAMAPK1GABRG2GABRB3
SCHEMBL2525793 0.74 MBOAT4 (0.34) ATRGAAMAPK1GABRG2GABRB3
SCHEMBL13647699 0.74 HCRTR1 (0.33) CASP6P2RX7
SCHEMBL12693213 0.73 NPC1 (0.46) MAPK1GABRG2GABRB3GABRA5
SCHEMBL2076032 0.71 EGLN2 (0.40) GAAMEN1KMT2A
SCHEMBL12215789 0.69 KDM5A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745052-B1 HIV INTEGRASE INHIBITORS: CYCLIC PYRIMIDINONE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2008-08-20 EP disclosed