SCHEMBL14101967

SCHEMBL14101967

COc1cc(OC)cc(-c2cc(-c3cc(N4CCCC4)ccc3C(F)(F)F)c(OCc3ccccc3)c3c2CCC3)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGDR2 Q9Y5Y4 4/20 0.34
TLR9 Q9NR96 4/20 0.34
TLR7 Q9NYK1 2/20 0.34
HTR6 P50406 2/20 0.33
AKR1B10 O60218 1/20 0.33
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720319 0.89 ITGB2 (0.36) S1PR1
SCHEMBL4720326 0.89 ITGB2 (0.36) S1PR1
SCHEMBL14101744 0.81 AKR1B10 (0.35) KDM4EALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL14101743 0.77 HTR2A (0.36) KDM4EALDH1A1MAPTL3MBTL1AKR1B10
SCHEMBL4720516 0.76 ITGB2 (0.35) S1PR1SOS1
SCHEMBL4720518 0.76 ITGB2 (0.35) S1PR1SOS1
SCHEMBL14102029 0.75 ACHE (0.40) KMT2AKDM4EALDH1A1MAPTL3MBTL1
SCHEMBL4720758 0.71 CDK1 (0.35) S1PR1SOS1
SCHEMBL4720760 0.71 CDK1 (0.35) S1PR1SOS1
SCHEMBL14102089 0.70 MAPT (0.36) MEN1KMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed