SCHEMBL14107168

SCHEMBL14107168

CC(=O)Oc1c(C)nc(S(C)(=O)=O)nc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.39
DPP4 P27487 2/20 0.37
DPP8 Q6V1X1 2/20 0.37
CDC7 O00311 1/20 0.37
DBF4 Q9UBU7 1/20 0.37
CNR1 P21554 8/20 0.37
ADRB3 P13945 1/20 0.37
GABRA1 P14867 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
OPRD1 P41143 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CNR2 P34972 4/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CRHR1 P34998 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4809317 0.89 ABCB11 (0.38) ABCB11CDC7DBF4CNR1ADRB3
SCHEMBL14107173 0.87 ABCB11 (0.41) ABCB11CNR1ADRB3GABRA1ADRA2B
SCHEMBL14107166 0.80 CRHR1 (0.40) DPP4DPP8CNR1MAPTKDM4E
SCHEMBL14107165 0.79 CYP3A4 (0.35) CNR1CNR2MAPTKMT2AKDM4E
SCHEMBL4804664 0.76 CNR1 (0.44) CNR1ADRB3GABRA1ADRA2BADRA2C
SCHEMBL4808908 0.75 CNR1 (0.42) CNR1ADRB3GABRA1ADRA2BADRA2C
SCHEMBL4810834 0.75 PTGS2 (0.42) DPP4CNR1ADRB3GABRA1ADRA2B
SCHEMBL4801796 0.73 CRHR1 (0.42) DPP4CNR1CNR2KDM4ECRHR1
SCHEMBL4809956 0.71 TDP1 (0.39) ABCB11CNR1CNR2MAPTKMT2A
SCHEMBL4809390 0.71 CNR1 (0.43) CNR1ADRB3GABRA1ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7405221-B2 Substituted pyrimidines MERCK & CO., INC. (US) 2008-07-29 US disclosed