SCHEMBL14128656

SCHEMBL14128656

CCOC(=O)C(F)(F)C1CCCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
HTT P42858 2/20 0.44
XBP1 P17861 1/20 0.44
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
USP2 O75604 1/20 0.42
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPK1 P28482 1/20 0.40
MAPK14 Q16539 1/20 0.40
FFAR1 O14842 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5530439 0.84 ESR1 (0.42) MAPK1TRPV1
SCHEMBL30276343 0.76 HTT (0.51) ALDH1A1HTTKMT2AMEN1TSHR
SCHEMBL2115724 0.74 ALDH1A1 (0.51) ALDH1A1HTTXBP1KMT2AKDM4E
SCHEMBL14825898 0.73 MAPK1 (0.42) ALDH1A1HTTXBP1KMT2AKDM4E
SCHEMBL30443664 0.72 MEN1 (0.41) KMT2AKDM4EMEN1TSHRLMNA
SCHEMBL9004030 0.72 IDO1 (0.49) ALDH1A1HTTKMT2AMEN1TSHR
SCHEMBL5468751 0.72 ALDH1A1 (0.49) ALDH1A1HTTXBP1KMT2AKDM4E
SCHEMBL61381 0.71 ALDH1A1 (0.63) ALDH1A1HTTKMT2AMEN1HPGD
SCHEMBL61382 0.71 ALDH1A1 (0.63) ALDH1A1HTTKMT2AMEN1HPGD
SCHEMBL6689518 0.71 KDM4E (0.46) ALDH1A1HTTXBP1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012163790-A1 SPIRO-[1,3]-OXAZINES AND SPIRO-[1,4]-OXAZEPINES AS BACE1 AND/OR BACE2 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-12-06 WO disclosed