SCHEMBL14134239

SCHEMBL14134239

Cc1ccc(-c2cnc(Nc3cccc(O)c3)o2)cc1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.66
FLT1 P17948 7/20 0.66
FLT4 P35916 7/20 0.66
VCP P55072 6/20 0.56
SIRT7 Q9NRC8 1/20 0.55
ALOX5 P09917 1/20 0.55
IMPDH2 P12268 2/20 0.51
DGAT1 O75907 1/20 0.48
TRPV1 Q8NER1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21311902 0.91 VCP (0.68) KDRFLT1FLT4VCPSIRT7
SCHEMBL21311878 0.86 VCP (0.64) KDRFLT1FLT4VCPSIRT7
SCHEMBL14057525 0.84 TRPV1 (0.66) KDRFLT1FLT4VCPSIRT7
SCHEMBL14058473 0.84 KDR (0.67) KDRFLT1FLT4VCPSIRT7
SCHEMBL1909825 0.81 KDR (0.49) KDRFLT1FLT4VCPSIRT7
SCHEMBL5184578 0.80 KDR (0.72) KDRFLT1FLT4VCPIMPDH2
Gw632046X SCHEMBL5475472 0.80 KDR (1.00) KDRFLT1FLT4VCPSIRT7
SCHEMBL14058062 0.78 IMPDH2 (0.66) KDRFLT1FLT4VCPSIRT7
SCHEMBL21311881 0.77 VCP (0.78) KDRFLT1FLT4VCPIMPDH2
SCHEMBL14134241 0.76 KDR (0.73) KDRFLT1FLT4SIRT7ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8865709-B2 Aminooxazole inhibitors of cyclin dependent kinases Neosome Life Sciences, LLC (US) 2014-10-21 US disclosed
US-20140051694-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases Neosome Life Sciences, LLC (US) 2014-02-20 US disclosed
US-8551992-B2 Aminooxazole inhibitors of cyclin dependent kinases Neosome Life Sciences, LLC (US) 2013-10-08 US disclosed
US-8546400-B2 1,3-Oxazole-4-carboxamides, 1,3-Thiazole-4-carboxamides, and 1,3-Imidazole-d-carboxamides as Inhibitors of cyclin Dependent kinases Neosome Life Sciences, LLC (US) 2013-10-01 US disclosed
US-20130184288-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases Neosome Life Sciences, LLC (US) 2013-07-18 US disclosed
US-20120302578-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases Neosome Life Sciences, LLC (US) 2012-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130184288-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases CDK1, CCNK, CCNI KDR 3471/4885FLT1 1646/4885FLT4 1762/4885
US-20120302578-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases CDK1, CCNK, CCNI KDR 3471/4885FLT1 1646/4885FLT4 1762/4885
US-20140051694-A1 Aminooxazole Inhibitors of Cyclin Dependent Kinases CDK1, CCNK, CCNI KDR 3471/4885FLT1 1646/4885FLT4 1762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.