SCHEMBL14154

SCHEMBL14154

Cc1ccc(C)c(CCCCN)c1

nearest known ligand 0.74

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.74
POLB P06746 2/20 0.42
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2A6 P11509 1/20 0.39
HTR2A P28223 2/20 0.39
HTR1D P28221 1/20 0.39
MAOA P21397 1/20 0.38
MPO P05164 1/20 0.36
TACR1 P25103 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10110932 0.98 TAAR1 (0.71) TAAR1POLBALDH1A1TDP1CYP1A2
SCHEMBL9469337 0.94 TAAR1 (0.77) TAAR1POLBALDH1A1TDP1CYP1A2
Hydrochloric Acid SCHEMBL21248269 0.92 TAAR1 (0.74) TAAR1POLBALDH1A1TDP1CYP1A2
SCHEMBL1869457 0.85 TAAR1 (1.00) TAAR1POLBALDH1A1TDP1CYP1A2
SCHEMBL8910791 0.84 TAAR1 (0.52) TAAR1CYP1A2CYP2A6HTR2AHTR1D
SCHEMBL11331960 0.82 TAAR1 (0.50) TAAR1CYP1A2CYP2A6HTR2AHTR1D
SCHEMBL11325501 0.82 TAAR1 (0.50) TAAR1CYP1A2CYP2A6HTR2AHTR1D
SCHEMBL11337231 0.82 TAAR1 (0.50) TAAR1CYP1A2CYP2A6HTR2AHTR1D
SCHEMBL11329871 0.82 TAAR1 (0.50) TAAR1CYP1A2CYP2A6HTR2AHTR1D
SCHEMBL11338772 0.82 TAAR1 (0.50) TAAR1CYP1A2CYP2A6HTR2AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9845297-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2017-12-19 US disclosed
US-20160031828-A1 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME SILICON VALLEY BANK 2016-02-04 US disclosed
US-9216979-B2 Antimicrobial compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2015-12-22 US disclosed
US-20130090326-A1 Antimicrobial Compounds and Methods of Making and Using the Same RIB-X PHARMACEUTICALS, INC. (US) 2013-04-11 US disclosed
WO-2011047323-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130090326-A1 Antimicrobial Compounds and Methods of Making and Using the Same MPO, LPO, CAT TAAR1 4463/4885POLB 525/4885ALDH1A1 1117/4885
US-20160031828-A1 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME MPO, LPO, CAT TAAR1 4463/4885POLB 525/4885ALDH1A1 1117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.