SCHEMBL14175652

SCHEMBL14175652

C=CC(=O)NCCc1c(Br)[nH]c2ccc(OC)cc12

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 0.76
MTNR1B P49286 15/20 0.76
NQO2 P16083 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP3A4 P08684 2/20 0.56
CYP2D6 P10635 2/20 0.56
CYP2C9 P11712 2/20 0.56
CYP2C19 P33261 2/20 0.56
TSHR P16473 1/20 0.56
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 2/20 0.55
HPGD P15428 2/20 0.55
HSD17B10 Q99714 2/20 0.55
POLB P06746 1/20 0.55
MDM2 Q00987 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1311849 0.86 MTNR1A (1.00) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL8946906 0.81 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2ALDH1A1KDM4E
SCHEMBL14175650 0.77 MTNR1A (0.76) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL3231477 0.77 MTNR1A (0.66) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL26989714 0.76 MTNR1A (0.80) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL8229569 0.74 HTR6 (0.72) MTNR1AMTNR1BCYP1A2TSHRALDH1A1
SCHEMBL8946916 0.73 MTNR1A (1.00) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL31543713 0.73 MTNR1A (1.00) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL31530479 0.73 MTNR1A (0.78) MTNR1AMTNR1BNQO2CYP1A2CYP3A4
SCHEMBL31530480 0.73 MTNR1A (0.78) MTNR1AMTNR1BNQO2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7381740-B2 Exert the beneficial effects of melatonin including anti-oxidation, sedation, anesthesia, protection of organs to chemical, infectious and cardiovascular damage, and can be administered in a water-based vehicle UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2008-06-03 US disclosed
US-7381740-B2 Exert the beneficial effects of melatonin including anti-oxidation, sedation, anesthesia, protection of organs to chemical, infectious and cardiovascular damage, and can be administered in a water-based vehicle UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2008-06-03 US disclosed