SCHEMBL14199075

SCHEMBL14199075

O=CCn1c(=O)oc2cc(O)ccc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MIF P14174 7/20 0.48
HPGD P15428 2/20 0.44
MAPK1 P28482 2/20 0.44
USP2 O75604 1/20 0.44
TSHR P16473 1/20 0.44
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
APEX1 P27695 1/20 0.40
CD74 P04233 2/20 0.40
SIGMAR1 Q99720 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
CBX7 O95931 1/20 0.39
CDYL Q9Y232 1/20 0.39
CDY1; CDY1B Q9Y6F8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14518249 0.81 MIF (0.65) MIFHPGDMAPK1USP2TSHR
SCHEMBL2757855 0.79 MIF (0.70) MIFMAPK1TSHRNPC1ALDH1A1
SCHEMBL14198763 0.78 MAPK1 (0.70) MIFHPGDMAPK1USP2TSHR
SCHEMBL3063571 0.78 LMNA (0.49) MIFHPGDKMT2AALDH1A1APEX1
SCHEMBL14199043 0.78 POLB (0.52) MIFHPGDKMT2AALDH1A1NPSR1
SCHEMBL14198915 0.76 KMO (0.49) ALDH1A1NPSR1
SCHEMBL14198929 0.76 NPC1 (0.39) MIFHPGDMAPK1USP2TSHR
SCHEMBL11218178 0.74 MIF (0.54) MIFHPGDMAPK1USP2TSHR
SCHEMBL14198758 0.72 IDO1 (0.66)
SCHEMBL14198764 0.72 MIF (0.65) MIFHPGDUSP2TSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-B1 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-05-07 EP disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed