SCHEMBL14199043

SCHEMBL14199043

COc1ccc2c(c1)oc(=O)n2CC=O

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.52
MET P08581 4/20 0.51
MAPT P10636 2/20 0.49
KMO O15229 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CDYL2 Q8N8U2 5/20 0.48
CDYL Q9Y232 5/20 0.48
CDY1; CDY1B Q9Y6F8 5/20 0.48
KMT2A Q03164 1/20 0.47
MIF P14174 3/20 0.47
CD74 P04233 2/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
TNIK Q9UKE5 2/20 0.46
CBX7 O95931 4/20 0.46
RECQL P46063 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5717564 0.86 MET (0.55) POLBMETMAPTKMOALDH1A1
SCHEMBL14518249 0.81 MIF (0.65) POLBALDH1A1HPGDKMT2AMIF
SCHEMBL8798927 0.80 MET (0.57) POLBMETMAPTKMOALDH1A1
Hydrochloric Acid SCHEMBL9157992 0.79 MET (0.56) POLBMETMAPTKMOALDH1A1
SCHEMBL4242148 0.79 KMO (0.61) POLBMETKMOCDYL2CDYL
SCHEMBL13140318 0.78 TP53 (0.58) POLBMETMAPTKMOALDH1A1
SCHEMBL2149713 0.78 MAPT (0.56) POLBMETMAPTKMOALDH1A1
SCHEMBL4413088 0.78 HPGD (0.59) POLBMETKMOHPGDCDYL2
SCHEMBL14199075 0.78 MIF (0.48) ALDH1A1HPGDNPSR1CDYLCDY1; CDY1B
SCHEMBL4228726 0.77 MAPT (0.58) POLBMETMAPTKMOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-B1 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-05-07 EP disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed