SCHEMBL14200488

SCHEMBL14200488

CCCC(C)N(C(=O)CC(C)(C)C)c1cccc(-c2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 1/20 0.39
COMT P21964 2/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
TP53 P04637 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.35
PTGES O14684 1/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
PTGS2 P35354 1/20 0.34
AOC3 Q16853 1/20 0.34
FFAR1 O14842 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200514 0.92 LTB4R2 (0.42) LTB4R2COMTNPC1RAB9ATP53
SCHEMBL14200490 0.90 LTB4R2 (0.38) LTB4R2COMTTP53SMN1; SMN2LMNA
SCHEMBL14200515 0.90 LTB4R2 (0.41) LTB4R2COMTNPC1RAB9ATP53
SCHEMBL14229354 0.86 TP53 (0.49) LTB4R2COMTNPC1RAB9ATP53
SCHEMBL14200476 0.85 LTB4R2 (0.44) LTB4R2COMTNPC1RAB9ATP53
SCHEMBL14200458 0.85 TAS1R3 (0.42) NPC1RAB9ATP53SMN1; SMN2LMNA
SCHEMBL14200493 0.85 LTB4R2 (0.40) LTB4R2TP53SMN1; SMN2LMNAHTT
SCHEMBL14200978 0.84 RIPK1 (0.39) NPC1RAB9ASMN1; SMN2LMNAHTT
SCHEMBL14200447 0.84 MAPK1 (0.36) SMN1; SMN2ALDH1A1HDAC8PTGS2
SCHEMBL14200443 0.84 ALDH1A1 (0.41) NPC1RAB9ASMN1; SMN2HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed