SCHEMBL14200871

SCHEMBL14200871

CCCCCC(C)N(C(=O)CC(C)(C)C)c1ccc(F)c(Br)c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.33
HDAC8 Q9BY41 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MMP2 P08253 2/20 0.31
MMP3 P08254 1/20 0.31
MLYCD O95822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200858 0.92 CYP1A2 (0.33) IDO1HDAC8CYP1A2CYP2D6CYP2C9
SCHEMBL14200495 0.88 RIPK1 (0.34) HDAC8POLBMLYCD
SCHEMBL14200885 0.88
SCHEMBL14201039 0.87 IDO1 (0.33) IDO1HDAC8CYP1A2CYP2D6CYP2C9
SCHEMBL14229738 0.87 CYP1A2 (0.33) IDO1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14201013 0.87 CYP1A2 (0.34) IDO1HDAC8CYP1A2CYP2D6CYP2C9
SCHEMBL14200485 0.87 ALDH1A1 (0.39) MEN1KMT2AMMP2MMP3
SCHEMBL14200981 0.85 CHRNA1 (0.35) CYP1A2CYP2C9CYP2C19KMT2AMMP2
SCHEMBL14201017 0.85 CYP1A2 (0.34) IDO1HDAC8CYP1A2CYP2D6CYP2C9
SCHEMBL14201033 0.82 IDO1 (0.33) IDO1HDAC8CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed