SCHEMBL14200877

SCHEMBL14200877

CCCN(CCC(C)(C)C)c1ncccc1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.41
AGTR2 P50052 1/20 0.41
AR P10275 2/20 0.39
HPGD P15428 4/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 1/20 0.36
ALDH1A1 P00352 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
CASP3 P42574 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200875 0.92 AGTR1 (0.48) AGTR1AGTR2ARHPGDCYP1A2
SCHEMBL14228976 0.85 AGTR1 (0.53) AGTR1AGTR2ARHPGDCYP1A2
SCHEMBL14228959 0.81 AGTR1 (0.54) AGTR1AGTR2ARHPGDCYP1A2
SCHEMBL14200700 0.80 HPGD (0.35) AGTR1AGTR2HPGDCYP1A2CYP2D6
SCHEMBL14200751 0.79 HPGD (0.37) AGTR1AGTR2HPGDCYP1A2CYP2D6
SCHEMBL5200518 0.78 KCNMA1 (0.47) AGTR1AGTR2HPGDCYP1A2CYP2D6
SCHEMBL14200874 0.74 AGTR1 (0.48) AGTR1AGTR2CYP1A2CYP2C9CYP2C19
SCHEMBL12125020 0.70 HPGD (0.43) AGTR1AGTR2HPGDCYP1A2CYP2D6
SCHEMBL6191221 0.69 HTT (0.45) HPGDCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL2526101 0.69 MAPT (0.39) ARALDH1A1L3MBTL1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed