SCHEMBL14202062

SCHEMBL14202062

Cc1ccc2c(c1)OCC(=O)N2Cc1cc(Cl)cc(N2CCNCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.47
BRD4 O60885 1/20 0.42
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
ADRB1 P08588 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
SLC5A1 P13866 3/20 0.41
SLC5A2 P31639 3/20 0.41
PIK3CG P48736 2/20 0.40
NMT1 P30419 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.39
HTR1A P08908 1/20 0.38
HTR3A P46098 1/20 0.38
DRD4 P21917 1/20 0.37
PLK1 P53350 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4477885 0.87 L3MBTL1 (0.52) HTR6BRD4CHRM2CHRM4ADRB1
SCHEMBL13973050 0.87 HTR6 (0.46) HTR6BRD4CHRM2CHRM4ADRB1
SCHEMBL4486014 0.74 POLB (0.57) HTR6CHRM2CHRM4ADRB1CHRM1
SCHEMBL4493695 0.74 HDAC1 (0.54) HTR6CHRM2CHRM4ADRB1CHRM1
SCHEMBL13960736 0.73 L3MBTL1 (0.48) BRD4SLC5A1SLC5A2L3MBTL1TSHR
SCHEMBL4674316 0.72 HTR6 (0.64) HTR6BRD4PIK3CGL3MBTL1TSHR
SCHEMBL13973049 0.71 SMN1; SMN2 (0.43) SLC5A1SLC5A2L3MBTL1HTT
SCHEMBL4678275 0.71 HTR6 (0.50) HTR6PIK3CGL3MBTL1DRD4
SCHEMBL8556616 0.71 TSHR (0.65) BRD4L3MBTL1TSHRDRD4
SCHEMBL4475776 0.71 L3MBTL1 (0.46) L3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603880-B1 QUINOLINONE/BENZOXAZINONE DERIVATIVES AND USES THEREOF HOFFMANN LA ROCHE (CH) 2008-05-07 EP disclosed