SCHEMBL14212432

SCHEMBL14212432

O=c1n(Cc2ccc(C(F)(F)F)nc2)nc2c(-c3ccc(OC(F)(F)F)cc3)c(-c3ccc(Cl)cc3)cnn12

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.80
CYP2C9 P11712 5/20 0.50
CYP2C19 P33261 5/20 0.50
CYP3A4 P08684 4/20 0.50
NR3C1 P04150 1/20 0.38
GPR139 Q6DWJ6 1/20 0.37
MALT1 Q9UDY8 2/20 0.37
CHRM5 P08912 1/20 0.36
PDE1B Q01064 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14211892 0.93 CNR1 (0.91) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14180828 0.92 CNR1 (0.66) CNR1CYP2C9CYP2C19CYP3A4GPR139
SCHEMBL14212437 0.92 CNR1 (0.80) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14211170 0.90 CNR1 (0.86) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14212434 0.90 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14181112 0.90 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14211173 0.90 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14181054 0.90 CNR1 (0.66) CNR1CYP2C9CYP2C19CYP3A4GPR139
SCHEMBL14212187 0.89 CNR1 (0.84) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL4798385 0.89 CNR1 (1.00) CNR1CYP2C9CYP2C19CYP3A4NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378418-B2 Azabicyclic heterocycles as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed
EP-1697370-B1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-04-25 EP disclosed