SCHEMBL14219655

SCHEMBL14219655

CONC(=O)c1cc(Cl)c(F)c(F)c1Nc1ncc(Br)cc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 7/20 0.38
PTGS2 P35354 1/20 0.36
MAP2K2 P36507 2/20 0.36
SMC2 O95347 1/20 0.36
EGFR P00533 1/20 0.36
CSNK2A2 P19784 1/20 0.36
SMC1A Q14683 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
Q6ZSR9 Q6ZSR9 1/20 0.36
BMP2K Q9NSY1 1/20 0.36
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PTK2 Q05397 2/20 0.33
S1PR3 Q99500 4/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
S1PR1 P21453 3/20 0.32
ABCB11 O95342 1/20 0.32
NQO2 P16083 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14222460 0.90 MAP2K1 (0.40) MAP2K1PTGS2MAP2K2SMC2EGFR
SCHEMBL14223057 0.89 MAP2K1 (0.41) MAP2K1MAP2K2SMC2EGFRCSNK2A2
SCHEMBL14222454 0.89 MAP2K1 (0.41) MAP2K1MAP2K2SMC2EGFRCSNK2A2
SCHEMBL14220164 0.87 PTGS2 (0.36) MAP2K1PTGS2MAP2K2SMC2EGFR
SCHEMBL14219660 0.87 MAP2K1 (0.50) MAP2K1MAP2K2SMC2EGFRCSNK2A2
SCHEMBL14219658 0.87 MAP2K1 (0.39) MAP2K1PTGS2MAP2K2SMC2EGFR
SCHEMBL14222462 0.87 ALDH1A1 (0.36) MAP2K1NPC1ALDH1A1S1PR3CSF1R
SCHEMBL14219689 0.85 DHODH (0.39) MAP2K1EGFRNPC1ALDH1A1S1PR3
SCHEMBL14220129 0.85 MAP2K1 (0.36) MAP2K1PTGS2MAP2K2SMC2EGFR
SCHEMBL14223218 0.84 MAP2K1 (0.48) MAP2K1MAP2K2SMC2EGFRCSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed