SCHEMBL14220129

SCHEMBL14220129

CONC(=O)c1cc(Cl)c(F)c(F)c1Nc1ncc(C)cc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 7/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 1/20 0.36
DHODH Q02127 3/20 0.36
PTGS2 P35354 1/20 0.34
MAP2K2 P36507 2/20 0.34
SMC2 O95347 1/20 0.34
EGFR P00533 1/20 0.34
CSNK2A2 P19784 1/20 0.34
SMC1A Q14683 1/20 0.34
AAK1 Q2M2I8 1/20 0.34
Q6ZSR9 Q6ZSR9 1/20 0.34
BMP2K Q9NSY1 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PTK2 Q05397 2/20 0.33
CSF1R P07333 1/20 0.32
CRHR1 P34998 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14222541 0.89 MAP2K1 (0.39) MAP2K1KDM4EMAPTDHODHMAP2K2
SCHEMBL14220128 0.89 PTGS2 (0.37) MAP2K1KDM4EMAPTDHODHPTGS2
SCHEMBL14219728 0.89 MAP2K1 (0.39) MAP2K1KDM4EMAPTDHODHMAP2K2
SCHEMBL14219718 0.87 DHODH (0.36) MAP2K1DHODHPTGS2MAP2K2SMC2
SCHEMBL14219719 0.87 MAP2K1 (0.48) MAP2K1MAP2K2SMC2EGFRCSNK2A2
SCHEMBL14223049 0.86 MAP2K1 (0.37) MAP2K1KDM4EMAPTDHODHMAP2K2
SCHEMBL14222457 0.85 DHODH (0.41) MAP2K1KDM4EMAPTDHODHEGFR
SCHEMBL14219655 0.85 MAP2K1 (0.38) MAP2K1MAPTPTGS2MAP2K2SMC2
SCHEMBL14220127 0.84 MAP2K1 (0.50) MAP2K1MAP2K2SMC2EGFRCSNK2A2
SCHEMBL14219650 0.84 MAP2K1 (0.50) MAP2K1MAP2K2SMC2EGFRCSNK2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041088-A2 N-HYDROXY BENZAMIDES WITH ANTITUMOR ACTIVITY EOS (ETHICAL ONCOLOGY SCIENCE) S.P.A. (IT) 2008-04-10 WO disclosed
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed