SCHEMBL14219657

SCHEMBL14219657

Bc1cnc(Nc2c(C(=O)NOCC=C)cc(Cl)c(F)c2F)c(C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
MAP2K1 Q02750 7/20 0.33
CSNK2A2 P19784 2/20 0.33
MAP2K2 P36507 2/20 0.33
SMC2 O95347 1/20 0.33
EGFR P00533 1/20 0.33
SMC1A Q14683 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
Q6ZSR9 Q6ZSR9 1/20 0.33
BMP2K Q9NSY1 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KAT6A Q92794 1/20 0.31
MAPK3 P27361 1/20 0.30
RAF1 P04049 1/20 0.30
PDGFRB P09619 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30
CSNK2A3 Q8NEV1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14220130 0.90 ALDH1A1 (0.37) ALDH1A1MAP2K1CSNK2A2MAP2K2SMC2
SCHEMBL14220157 0.90 MEN1 (0.42) ALDH1A1MAP2K1MAP2K2MEN1KMT2A
SCHEMBL14219727 0.88 MEN1 (0.34) MAP2K1CSNK2A2MAP2K2SMC2EGFR
SCHEMBL14219716 0.87 ALDH1A1 (0.36) ALDH1A1MAP2K1CSNK2A2MAP2K2SMC2
SCHEMBL14220164 0.86 PTGS2 (0.36) MAP2K1CSNK2A2MAP2K2SMC2EGFR
SCHEMBL14219659 0.84 MAP2K1 (0.44) MAP2K1CSNK2A2MAP2K2SMC2EGFR
SCHEMBL14223049 0.83 MAP2K1 (0.37) ALDH1A1MAP2K1CSNK2A2MAP2K2SMC2
SCHEMBL14219743 0.83 MEN1 (0.42) ALDH1A1MAP2K1CSNK2A2MAP2K2SMC2
SCHEMBL14223224 0.81 ALDH1A1 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL14222456 0.81 DHODH (0.39) MAP2K1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed