SCHEMBL14220130

SCHEMBL14220130

C=CCONC(=O)c1cc(Cl)c(F)c(F)c1Nc1ncc(C)cc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAP2K1 Q02750 7/20 0.34
CSNK2A2 P19784 2/20 0.34
MAP2K2 P36507 2/20 0.34
SMC2 O95347 1/20 0.34
EGFR P00533 1/20 0.34
SMC1A Q14683 1/20 0.34
AAK1 Q2M2I8 1/20 0.34
Q6ZSR9 Q6ZSR9 1/20 0.34
BMP2K Q9NSY1 1/20 0.34
LCK P06239 1/20 0.32
DHODH Q02127 1/20 0.32
TXK P42681 1/20 0.32
JAK3 P52333 1/20 0.32
BTK Q06187 1/20 0.32
ITK Q08881 1/20 0.32
KAT6A Q92794 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14219657 0.90 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ATDP1MAP2K1
SCHEMBL14219716 0.90 ALDH1A1 (0.36) ALDH1A1MEN1KMT2ATDP1MAP2K1
SCHEMBL14223049 0.90 MAP2K1 (0.37) ALDH1A1MEN1KMT2ATDP1MAP2K1
SCHEMBL14220117 0.85 MEN1 (0.51) MEN1KMT2ATDP1MAP2K1CSNK2A2
SCHEMBL14219743 0.84 MEN1 (0.42) ALDH1A1MEN1KMT2ATDP1MAP2K1
SCHEMBL14219843 0.84 MAP2K1 (0.45) MAP2K1CSNK2A2MAP2K2SMC2EGFR
SCHEMBL14223052 0.84 MAP2K1 (0.45) MAP2K1CSNK2A2MAP2K2SMC2EGFR
SCHEMBL14219656 0.83 PTGS2 (0.41) MEN1KMT2ATDP1MAP2K1CSNK2A2
SCHEMBL14223224 0.82 ALDH1A1 (0.44) ALDH1A1MEN1KMT2APOLB
SCHEMBL14219853 0.81 MAP2K1 (0.40) ALDH1A1MEN1KMT2ATDP1MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041088-A2 N-HYDROXY BENZAMIDES WITH ANTITUMOR ACTIVITY EOS (ETHICAL ONCOLOGY SCIENCE) S.P.A. (IT) 2008-04-10 WO disclosed
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed