SCHEMBL14219679

SCHEMBL14219679

Cc1cc(Br)cnc1Nc1c(C(=O)O)ccc(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 6/20 0.46
MAP2K2 P36507 2/20 0.46
DHODH Q02127 8/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
SORT1 Q99523 3/20 0.38
S1PR3 Q99500 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14219621 0.88 MAP2K1 (0.48) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14219608 0.86 DHODH (0.54) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14222530 0.86 NPC1 (0.40) MAP2K1DHODHNPC1ALDH1A1LMNA
SCHEMBL14219680 0.85 MAP2K1 (0.55) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14220139 0.84 NPC1 (0.38) MAP2K1DHODHNPC1ALDH1A1LMNA
SCHEMBL14223198 0.83 MAP2K1 (0.46) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14219682 0.82 MAP2K1 (0.44) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14219689 0.82 DHODH (0.39) MAP2K1DHODHNPC1ALDH1A1LMNA
SCHEMBL14219811 0.81 MAP2K1 (0.44) MAP2K1MAP2K2DHODHLMNAGAA
SCHEMBL14220152 0.81 MAP2K1 (0.63) MAP2K1MAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041088-A2 N-HYDROXY BENZAMIDES WITH ANTITUMOR ACTIVITY EOS (ETHICAL ONCOLOGY SCIENCE) S.P.A. (IT) 2008-04-10 WO disclosed
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed