SCHEMBL14220139

SCHEMBL14220139

Cc1cc(Br)cnc1Nc1c(C(=O)O)cc(Br)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
DHODH Q02127 6/20 0.36
MAP2K1 Q02750 1/20 0.34
SORT1 Q99523 3/20 0.34
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
GABRA4 P48169 1/20 0.33
GABRE P78334 1/20 0.33
GABRA6 Q16445 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14222530 0.90 NPC1 (0.40) NPC1ALDH1A1LMNAGAADHODH
SCHEMBL14219689 0.88 DHODH (0.39) NPC1ALDH1A1LMNAGAADHODH
SCHEMBL14220106 0.88 DHODH (0.46) LMNAGAADHODHMAP2K1SORT1
SCHEMBL14219688 0.88 LMNA (0.36) LMNAGAADHODHMAP2K1GABRP
SCHEMBL14219679 0.84 MAP2K1 (0.46) NPC1ALDH1A1LMNAGAADHODH
SCHEMBL14219814 0.84 DHODH (0.43) LMNAGAADHODHMAP2K1SORT1
SCHEMBL14219822 0.81 DHODH (0.38) LMNAGAADHODHMAP2K1
SCHEMBL14219622 0.81 MAP2K1 (0.47) MAP2K1EGFR
SCHEMBL14219723 0.80 MAP2K1 (0.39) NPC1ALDH1A1MAP2K1EGFRMEN1
SCHEMBL14219677 0.80 DHODH (0.39) DHODHMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed