SCHEMBL14220128

SCHEMBL14220128

Cc1cnc(Nc2c(C(=O)NOC(C)(C)C)cc(Cl)c(F)c2F)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
SMC2 O95347 1/20 0.33
EGFR P00533 1/20 0.33
CSNK2A2 P19784 1/20 0.33
MAP2K2 P36507 1/20 0.33
MAP2K1 Q02750 1/20 0.33
SMC1A Q14683 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
Q6ZSR9 Q6ZSR9 1/20 0.33
BMP2K Q9NSY1 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
DHODH Q02127 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14219656 0.90 PTGS2 (0.41) PTGS2SMC2EGFRCSNK2A2MAP2K2
SCHEMBL14223203 0.90 KDM4E (0.36) PTGS2KDM4EMAPTEGFRMAP2K2
SCHEMBL14220129 0.89 MAP2K1 (0.36) PTGS2KDM4EMAPTSMC2EGFR
SCHEMBL14219728 0.86 MAP2K1 (0.39) KDM4EMAPTSMC2EGFRCSNK2A2
SCHEMBL14219719 0.84 MAP2K1 (0.48) SMC2EGFRCSNK2A2MAP2K2MAP2K1
SCHEMBL14223049 0.83 MAP2K1 (0.37) KDM4EMAPTSMC2EGFRCSNK2A2
SCHEMBL14222457 0.83 DHODH (0.41) KDM4EMAPTEGFRMAP2K1DHODH
SCHEMBL14220127 0.81 MAP2K1 (0.50) SMC2EGFRCSNK2A2MAP2K2MAP2K1
SCHEMBL14219650 0.81 MAP2K1 (0.50) SMC2EGFRCSNK2A2MAP2K2MAP2K1
SCHEMBL14219845 0.80 MAP2K2 (0.35) PTGS2MAP2K2MAP2K1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041088-A2 N-HYDROXY BENZAMIDES WITH ANTITUMOR ACTIVITY EOS (ETHICAL ONCOLOGY SCIENCE) S.P.A. (IT) 2008-04-10 WO disclosed
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed