SCHEMBL14224513

SCHEMBL14224513

Cc1ccc(CNC(=O)C[S+](C)[O-])c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 1/20 0.42
P2RX7 Q99572 9/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
ERCC1 P07992 1/20 0.40
ERCC4 Q92889 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
EPHX2 P34913 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1989133 0.88 ALDH1A1 (0.41) ALDH1A1P2RX7NPC1RAB9AERCC1
SCHEMBL14197092 0.83 NPC1 (0.40) KMT2ALMNAALDH1A1P2RX7NPC1
SCHEMBL14224512 0.78 KMT2A (0.49) KMT2ALMNAALDH1A1P2RX7ERCC1
SCHEMBL14224535 0.77 LMNA (0.52) KMT2ALMNAALDH1A1P2RX7NPC1
SCHEMBL18251699 0.75 ALDH1A1 (0.48) KMT2ALMNAALDH1A1P2RX7NPC1
SCHEMBL1871724 0.71 EPHX2 (0.42) P2RX7EPHX2
SCHEMBL18585814 0.69 APOBEC3A (0.53) KMT2ALMNAALDH1A1NPC1RAB9A
SCHEMBL14224777 0.69 GAA (0.49) KMT2AALDH1A1P2RX7NPC1RAB9A
SCHEMBL24776466 0.68 SLC6A4 (0.50) ALDH1A1
SCHEMBL30435098 0.68 SLC6A4 (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7354919-B2 Isoxazole compositions useful as inhibitors of ERK VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-04-08 US disclosed